SCHEMBL5048134

SCHEMBL5048134

COC(=O)c1c(C#N)ccn1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
GAA P10253 2/20 0.37
DAPK3 O43293 1/20 0.37
JAK2 O60674 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
ABL1 P00519 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
PDGFRA P16234 1/20 0.37
PRKACA P17612 1/20 0.37
LTK P29376 1/20 0.37
GRK5 P34947 1/20 0.37
KDR P35968 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
CSNK1A1 P48729 1/20 0.37
CDK8 P49336 1/20 0.37
CLK2 P49760 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2446096 0.75 DAPK3 (0.41) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL4247977 0.74 ABL1 (0.40) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL13731286 0.74 DAPK3 (0.40) ALDH1A1DAPK3JAK2PRKD3MAP4K4
Hydrochloric Acid SCHEMBL1396143 0.72 ABL1 (0.39) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL20101952 0.71 ALDH1A1 (0.40) ALDH1A1GAADAPK3JAK2PRKD3
Ethane SCHEMBL15559374 0.71 ABL1 (0.38) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL31294085 0.70 NOTUM (0.43) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL3938677 0.69 KDM4E (0.45) ALDH1A1GAAKDM4EMAPTRXFP1
SCHEMBL16007133 0.69 ALDH1A1 (0.47) ALDH1A1GAADAPK3JAK2PRKD3
SCHEMBL26301302 0.68 DAPK3 (0.35) ALDH1A1GAADAPK3JAK2PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966215-A1 CONDENSED HETEROCYCLIC COMPOUNDS USEFUL AS DPP-IV INHIBITORS Novartis AG (CH) 2008-09-10 EP disclosed
WO-2007071738-A1 CONDENSED HETEROCYCLIC COMPOUNDS USEFUL AS DPP-IV INHIBITORS NOVARTIS AG (CH) 2007-06-28 WO disclosed