SCHEMBL5048385

SCHEMBL5048385

COc1cc(N2CCN(CC(C)C(N)C=O)CC2)c(Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.41
ADRA1A P35348 3/20 0.37
ADRA1B P35368 3/20 0.37
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
ADRA1D P25100 2/20 0.37
MAPT P10636 4/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR7 P34969 2/20 0.36
HTR1A P08908 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5051976 0.99 CCR1 (0.41) CCR1ADRA1AADRA1BADRB2ADRB1
SCHEMBL5048319 0.74 IGF1R (0.49) ADRB1MAPTALDH1A1LMNAMAPK1
SCHEMBL4501206 0.73 NPSR1 (0.48) CCR1MAPTALDH1A1LMNAKDM4E
SCHEMBL4501202 0.73 NPSR1 (0.48) CCR1MAPTALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL4502722 0.72 NPSR1 (0.48) CCR1MAPTALDH1A1LMNAKDM4E
SCHEMBL3223360 0.70 ALDH1A1 (0.47) CCR1MAPTALDH1A1LMNAMAPK1
SCHEMBL4074344 0.70 CCR1 (0.47) CCR1MAPTALDH1A1LMNAMAPK1
SCHEMBL19175191 0.66 CHRM1 (0.48) MAPTKDM4EMEN1KMT2ACHRM5
SCHEMBL2874775 0.66 HTR3A (0.60) ADRB1MAPTLMNAHTR7HTR1A
SCHEMBL3227831 0.65 CCR1 (0.49) CCR1MAPTKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973880-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Brystol-Myers Squibb Company (US) 2008-10-01 EP disclosed
WO-2007087585-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-02 WO disclosed