SCHEMBL5048864

SCHEMBL5048864

CCCCCCCCCCCCNC(=O)c1cccc(CNCc2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.62
POLB P06746 1/20 0.62
MRGPRX4 Q96LA9 2/20 0.57
TP53BP1 Q12888 1/20 0.57
HDAC3 O15379 2/20 0.55
HDAC1 Q13547 2/20 0.55
HDAC2 Q92769 1/20 0.55
NAMPT P43490 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MLYCD O95822 2/20 0.53
NAAA Q02083 1/20 0.52
MEN1 O00255 1/20 0.52
PLA2G1B P04054 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
GAA P10253 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852697 0.92 MLYCD (0.58) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL5044022 0.92 MRGPRX4 (0.56) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL2358408 0.88 POLB (0.80) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL5044055 0.88 MLYCD (0.51) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL5043673 0.88 ALDH1A1 (0.50) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL7220582 0.87 POLB (0.82) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL1855176 0.86 NAAA (0.68) HDAC3HDAC1HDAC2SMN1; SMN2MLYCD
SCHEMBL1853372 0.86 ALDH1A1 (0.56) ALDH1A1POLBMRGPRX4TP53BP1HDAC3
SCHEMBL27619583 0.84 SMN1; SMN2 (0.58) HDAC3NAMPTSMN1; SMN2MLYCDNAAA
SCHEMBL5044180 0.83 MRGPRX4 (0.48) ALDH1A1POLBMRGPRX4TP53BP1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed