SCHEMBL5049330

SCHEMBL5049330

CCCCCCCCNC(=O)c1cccc(-c2ccc(C[CH]c3ccc(C(F)(F)F)cc3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
NAAA Q02083 2/20 0.47
MRGPRX4 Q96LA9 1/20 0.47
MLYCD O95822 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45
TP53BP1 Q12888 1/20 0.44
ERN1 O75460 1/20 0.43
HDAC3 O15379 1/20 0.43
NAMPT P43490 2/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
EPHX2 P34913 1/20 0.42
BCL2L1 Q07817 1/20 0.42
MCL1 Q07820 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
AKR1C3 P42330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5046329 1.00 ALDH1A1 (0.48) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL5047208 0.88 AKR1C3 (0.47) ALDH1A1POLBHDAC1EPHX2AKR1C3
SCHEMBL5044168 0.83 ALDH1A1 (0.47) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL5045562 0.83 ALDH1A1 (0.47) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL1861375 0.81 NAAA (0.48) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL1857017 0.81 NAAA (0.48) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL5046272 0.81 NAAA (0.57) NAAAMLYCDSMN1; SMN2HDAC1HDAC2
SCHEMBL5039647 0.80 TACR1 (0.54) HDAC2EPHX2BCL2L1MCL1AKR1C3
SCHEMBL5047162 0.78 HDAC1 (0.44) ALDH1A1POLBNAAAMRGPRX4MLYCD
SCHEMBL5039660 0.78 HDAC1 (0.44) ALDH1A1POLBNAAAMRGPRX4MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed