SCHEMBL5039660

SCHEMBL5039660

CCCCCCCCNC(=O)c1cccc(-c2ccc(CC(NC(=O)C(=O)O)c3ccc(C(F)(F)F)cc3)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
NAAA Q02083 1/20 0.44
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.42
KIFC1 Q9BW19 6/20 0.42
MLYCD O95822 1/20 0.41
PTGS2 P35354 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
TP53BP1 Q12888 1/20 0.40
PTPN1 P18031 1/20 0.40
BCL2L1 Q07817 1/20 0.40
MCL1 Q07820 1/20 0.40
EPHX2 P34913 1/20 0.40
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047162 1.00 HDAC1 (0.44) HDAC1HDAC2NAAAALDH1A1POLB
SCHEMBL1852984 0.90 MLYCD (0.51) NAAAALDH1A1MLYCDSMN1; SMN2EPHX2
SCHEMBL1853396 0.85 MLYCD (0.47) NAAAALDH1A1POLBMRGPRX4MLYCD
SCHEMBL5045562 0.85 ALDH1A1 (0.47) HDAC1HDAC2NAAAALDH1A1POLB
SCHEMBL5044168 0.85 ALDH1A1 (0.47) HDAC1HDAC2NAAAALDH1A1POLB
SCHEMBL5039508 0.82 ROCK2 (0.44) HDAC1NAAAKIFC1MLYCDPTGS2
SCHEMBL1861375 0.80 NAAA (0.48) HDAC1HDAC2NAAAALDH1A1POLB
SCHEMBL1857017 0.80 NAAA (0.48) HDAC1HDAC2NAAAALDH1A1POLB
SCHEMBL5046973 0.78 UTS2R (0.47) SMN1; SMN2EPHX2PPARGPPARAMME
SCHEMBL4978882 0.78 PLK1 (0.47) HDAC1SMN1; SMN2PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP disclosed