SCHEMBL5053380

SCHEMBL5053380

CCP(=O)(Cl)N(C#N)N(C(C)C)C(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8719762 0.68 TP53 (0.31)
SCHEMBL28117340 0.59 TRPM8 (0.33)
SCHEMBL8919030 0.59 TSHR (0.31)
SCHEMBL28295068 0.56 MEN1 (0.38)
SCHEMBL15875801 0.54
SCHEMBL25062104 0.54 FDPS (0.37)
SCHEMBL11020160 0.54 TSHR (0.33)
SCHEMBL642627 0.53
SCHEMBL11871347 0.52
SCHEMBL9419924 0.51

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075549-B1 ELECTRONIC METHODS FOR THE DETECTION OF ANALYTES UTILIZING MONOLAYERS CLINICAL MICRO SENSORS INC (US) 2008-09-03 EP disclosed
US-7090804-B2 Amplification of nucleic acids with electronic detection CLINICAL MIRCO SENSORS, INC. (US) 2006-08-15 US disclosed
WO-2001006016-A9 AMPLIFICATION OF NUCLEIC ACIDS WITH ELECTRONIC DETECTION CLINICAL MICRO SENSORS INC (US) 2002-07-11 WO disclosed
EP-1194593-A2 AMPLIFICATION OF NUCLEIC ACIDS WITH ELECTRONIC DETECTION Clinical Micro Sensors, Inc. (US) 2002-04-10 EP disclosed
US-20020006643-A1 Screening sample for target nucleotide sequences; hybridize primer, incubate with enzyme, dissociate hybridization complex, detect electron transfer between electrode transfer particle OSMETECH TECHNOLOGY, INC. 2002-01-17 US disclosed
EP-1075549-A1 ELECTRONIC METHODS FOR THE DETECTION OF ANALYTES UTILIZING MONOLAYERS Clinical Micro Sensors, Inc. (US) 2001-02-14 EP disclosed
EP-1075541-A1 ELECTRONIC DETECTION OF NUCLEIC ACIDS USING MONOLAYERS Clinical Micro Sensors (US) 2001-02-14 EP disclosed
WO-2001006016-A2 AMPLIFICATION OF NUCLEIC ACIDS WITH ELECTRONIC DETECTION CLINICAL MICRO SENSORS, INC. (US) 2001-01-25 WO disclosed
EP-1051517-A2 AMPLIFICATION OF NUCLEIC ACIDS WITH ELECTRONIC DETECTION Clinical Micro Sensors, Inc. (US) 2000-11-15 EP disclosed
WO-1999057317-A9 ELECTRONIC METHODS FOR THE DETECTION OF ANALYTES UTILIZING MONOLAYERS CLINICAL MICRO SENSORS INC (US) 2000-02-17 WO disclosed
WO-1999057319-A1 ELECTRONIC DETECTION OF NUCLEIC ACIDS USING MONOLAYERS CLINICAL MICRO SENSORS (US) 1999-11-11 WO disclosed
WO-1999057317-A1 ELECTRONIC METHODS FOR THE DETECTION OF ANALYTES UTILIZING MONOLAYERS CLINICAL MICRO SENSORS, INC. (US) 1999-11-11 WO disclosed
WO-1999037819-A2 AMPLIFICATION OF NUCLEIC ACIDS WITH ELECTRONIC DETECTION CLINICAL MICRO SENSORS, INC. (US) 1999-07-29 WO disclosed