SCHEMBL5059161

SCHEMBL5059161

O=C(CN1CCNCCNCCNCC1)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.53
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
SIGMAR1 Q99720 2/20 0.50
MAPK1 P28482 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 1/20 0.48
ITGB3 P05106 2/20 0.47
ITGA2B P08514 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
GLA P06280 1/20 0.45
HTR2C P28335 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43
HTR1A P08908 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL28444822 0.99 EGFR (0.52) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL6601404 0.98 EGFR (0.54) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL25421283 0.97 EGFR (0.53) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
Hydrochloric Acid SCHEMBL21814218 0.97 EGFR (0.56) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL3422030 0.97 EGFR (0.53) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
Bromide SCHEMBL14247934 0.96 EGFR (0.52) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL10317072 0.93 ALDH1A1 (0.54) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL25134221 0.93 EGFR (0.50) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL17921386 0.91 EGFR (0.48) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1
SCHEMBL5054607 0.91 EGFR (0.48) EGFRALDH1A1SMN1; SMN2SIGMAR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001052899-A1 CHELATING AGENTS AND METHOD FOR THEIR USE AS TANDEM METAL CHELATORS AND HYDROPHILIC SPACERS FOR MEDICAL DIAGNOSIS AND THERAPY MALLINCKRODT INC. (US) 2001-07-26 WO claimed
EP-2495563-A1 DIAGNOSTIC AGENT FOR INFECTIOUS DISEASES Fujifilm RI Pharma Co., Ltd. (JP) 2012-09-05 EP disclosed
US-20120219500-A1 DIAGNOSTIC AGENT FOR INFECTIOUS DISEASES FUJIFILM RI PHARMA CO., LTD. (JP) 2012-08-30 US disclosed
WO-2008144728-A1 CONJUGATES WHICH BIND A BLOOD PROTEIN SUCH AS HUMAN SERUM ALBUMIN AND METHODS OF USING THE SAME IN DIAGNOSTIC AND THERAPEUTIC APPLICATIONS BRACCO IMAGING S.P.A. (IT) 2008-11-27 WO disclosed
US-20080181847-A1 Targeted Imaging and/or Therapy Using the Staudinger Ligation KONINKLIJKE PHILIPS ELECTRONICS, N.V. (NL) 2008-07-31 US disclosed
US-20080181847-A1 Targeted Imaging and/or Therapy Using the Staudinger Ligation KONINKLIJKE PHILIPS ELECTRONICS, N.V. (NL) 2008-07-31 US disclosed
US-20080124270-A1 Compounds Useful as Metal Chelators BRACCO IMAGING S.P.A. (IT) 2008-05-29 US disclosed
US-20080124270-A1 Compounds Useful as Metal Chelators BRACCO IMAGING S.P.A. (IT) 2008-05-29 US disclosed
US-20080124270-A1 Compounds Useful as Metal Chelators BRACCO IMAGING S.P.A. (IT) 2008-05-29 US disclosed
US-20070167615-A1 Macrocyclic oligonucleotide labeling reactants and conjugates derived thereof WALLAC OY (FI) 2007-07-19 US disclosed
US-20070167615-A1 Macrocyclic oligonucleotide labeling reactants and conjugates derived thereof WALLAC OY (FI) 2007-07-19 US disclosed
EP-1699466-A2 NEW COMPOUNDS USEFUL AS METAL CHELATORS Bracco Imaging, S.P.A. (IT) 2006-09-13 EP disclosed
WO-2005062828-A2 NEW COMPOUNDS USEFUL AS METAL CHELATORS BRACCO IMAGING S.P.A. (IT) 2005-07-14 WO disclosed
WO-2001052898-A9 METHODS FOR INCORPORATING METAL CHELATORS AT CARBOXYL-TERMINAL SITE OF PEPTIDES MALLINCKRODT INC (US) 2002-10-31 WO disclosed
WO-2001052898-A1 METHODS FOR INCORPORATING METAL CHELATORS AT CARBOXYL-TERMINAL SITE OF PEPTIDES MALLINCKRODT INC. (US) 2001-07-26 WO disclosed
WO-2001052900-A2 NOVEL ORTHOGONALLY PROTECTED AMINO ACID CHELATORS FOR BIOMEDICAL APPLICATIONS MALLINCKRODT INC. (US) 2001-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080181847-A1 Targeted Imaging and/or Therapy Using the Staudinger Ligation BTD, HLCS, BOLA2; BOLA2B EGFR 689/4885ALDH1A1 1007/4885SMN1; SMN2 2929/4885
US-20070167615-A1 Macrocyclic oligonucleotide labeling reactants and conjugates derived thereof POLRMT, RTCB, POLM EGFR 792/4885ALDH1A1 2550/4885SMN1; SMN2 2654/4885
US-20080124270-A1 Compounds Useful as Metal Chelators PAICS, PHOSPHO1, PPIP5K2 EGFR 3022/4885ALDH1A1 4035/4885SMN1; SMN2 3701/4885
US-20120219500-A1 DIAGNOSTIC AGENT FOR INFECTIOUS DISEASES NISCH, CNDP2, MYADM EGFR 4518/4885ALDH1A1 1641/4885SMN1; SMN2 2683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.