SCHEMBL5063200

SCHEMBL5063200

CC(C)(C)OC(=O)NC(CC(=O)O)Cc1cccc(Br)c1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.62
CTSK P43235 5/20 0.62
CTSB P07858 3/20 0.62
ATM Q13315 1/20 0.54
CTSL P07711 2/20 0.46
APP P05067 4/20 0.45
AAK1 Q2M2I8 4/20 0.45
ACE P12821 1/20 0.45
KLK5 Q9Y337 1/20 0.44
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4860365 1.00 CTSS (0.62) CTSSCTSKCTSBATMCTSL
SCHEMBL30597876 1.00 CTSS (0.62) CTSSCTSKCTSBATMCTSL
SCHEMBL4598553 0.89 CTSS (0.58) CTSSCTSKCTSBATMCTSL
SCHEMBL4859984 0.88 CTSS (0.61) CTSSCTSKCTSBATMCTSL
SCHEMBL4859989 0.88 CTSS (0.61) CTSSCTSKCTSBATMCTSL
SCHEMBL31758020 0.87 ATM (0.55) CTSSCTSKCTSBATMCTSL
SCHEMBL489490 0.86 ATM (0.70) CTSSCTSKCTSBATMCTSL
SCHEMBL489489 0.86 ATM (0.70) CTSSCTSKCTSBATMCTSL
SCHEMBL1519945 0.86 ATM (0.70) CTSSCTSKCTSBATMCTSL
SCHEMBL742226 0.86 CTSL (0.62) CTSSCTSKCTSBATMCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486762-A Novel compound and use method and application thereof 中国医学科学院医药生物技术研究所 2024-02-02 CN disclosed
CN-116693414-A Compound with 3CL protease inhibition activity and application thereof 深圳市小分子新药创新中心有限公司 2023-09-05 CN disclosed
US-20080306040-A1 Antibacterial amide macrocycles VII AICURIS GMBH & CO. KG (DE) 2008-12-11 US disclosed
US-20080306040-A1 Antibacterial amide macrocycles VII AICURIS GMBH & CO. KG (DE) 2008-12-11 US disclosed
US-20080306040-A1 Antibacterial amide macrocycles VII AICURIS GMBH & CO. KG (DE) 2008-12-11 US disclosed
WO-2007006548-A2 ANTIBACTERIAL AMIDE MACROCYCLES VII AICURIS GMBH & CO. KG (DE) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306040-A1 Antibacterial amide macrocycles VII AADAC, AAAS, NOD2 CTSS 88/4885CTSK 93/4885CTSB 60/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.