SCHEMBL5064901

SCHEMBL5064901

Nc1nc(N)c(-c2ccccc2)c(S(N)(=O)=O)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.50
HEXA P06865 1/20 0.50
HEXB P07686 1/20 0.50
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
CA7 P43166 1/20 0.47
ADORA2A P29274 3/20 0.41
ADORA1 P30542 3/20 0.41
POLB P06746 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2B P29275 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162150 0.79 DHFR (0.66) DHFRHEXAHEXBADORA2AADORA1
SCHEMBL5064900 0.72 ADORA1 (0.50) DHFRCA12CA1CA2CA9
SCHEMBL2187724 0.72 CA1 (0.48) CA12CA1CA2CA9CA7
SCHEMBL2473930 0.72 DHFR (0.58) DHFRHEXAHEXBADORA2AADORA1
SCHEMBL3500167 0.71 DHFR (0.61) DHFRHEXAHEXBADORA2AKDM4E
SCHEMBL1031028 0.71 DHFR (0.56) DHFRHEXAHEXBADORA2AADORA1
Hydrochloric Acid SCHEMBL15487768 0.71 DHFR (0.56) DHFRHEXAHEXBADORA2AADORA1
SCHEMBL12495983 0.67 ADORA2A (0.52) DHFRHEXAHEXBADORA2AADORA1
SCHEMBL7256603 0.67 DHFR (0.47) DHFRHEXAHEXBADORA2AADORA1
SCHEMBL3498787 0.67 HEXA (1.00) DHFRHEXAHEXBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008079907-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY RIGEL PHARMACEUTICALS, INC. (US) 2008-07-03 WO claimed