SCHEMBL5067014

SCHEMBL5067014

CCOC(=O)Cc1cc(N)ccc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAOA P21397 1/20 0.46
MAPK1 P28482 1/20 0.44
PKM P14618 1/20 0.43
PPIB P23284 1/20 0.42
PPIA P62937 1/20 0.42
PPID Q08752 1/20 0.42
PPIG Q13427 1/20 0.42
ALDH1A1 P00352 4/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
SHMT2 P34897 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
EGFR P00533 2/20 0.41
NLRP3 Q96P20 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9081693 0.88 LMNA (0.47) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL13564344 0.87 LMNA (0.46) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL2194027 0.85 EGFR (0.56) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL502012 0.85 ALDH1A1 (0.45) LMNAMAPK1ALDH1A1MAPTHPGD
SCHEMBL4277534 0.84 MAOA (0.44) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL3720048 0.84 LMNA (0.44) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL2131319 0.83 LMNA (0.46) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL27459157 0.83 NLRP3 (0.53) CYP1A2MAPK1PKMALDH1A1MAPT
SCHEMBL15835741 0.83 LMNA (0.50) LMNACYP1A2CYP3A4MAOAMAPK1
SCHEMBL2190989 0.83 DPP4 (0.49) LMNACYP1A2CYP3A4MAOAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120289540-A1 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES DECIPHERA PHARMACEUTICALS, LLC (US) 2012-11-15 US disclosed
US-8188113-B2 For example, 1-(5-(2-amino-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)-2-fluorophenyl)-3-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)urea; for treatment of mammalian cancers and inflammatory diseases including rheumatoid arthritis, retinopathies DECIPHERA PHARMACEUTICALS, INC. (US) 2012-05-29 US disclosed
CN-101553232-A Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS LLC (US) 2009-10-07 CN disclosed
US-20080114006-A1 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PARMACEUTICALS, LLC (US) 2008-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120289540-A1 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES BRAF, PRKDC, RAF1 LMNA 3483/4885CYP1A2 3849/4885CYP3A4 3505/4885
US-20080114006-A1 Kinase inhibitors useful for the treatment of proliferative diseases BRAF, PRKDC, RAF1 LMNA 3483/4885CYP1A2 3849/4885CYP3A4 3505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.