SCHEMBL5067796

SCHEMBL5067796

CSCC[C@H](N)C(=O)c1ccc([C](c2ccccc2)c2ccccc2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PKM P14618 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
KMO O15229 2/20 0.36
TSHR P16473 1/20 0.35
CCR1 P32246 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
RAB9A P51151 2/20 0.34
MARS1 P56192 2/20 0.34
NPC1 O15118 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CRHBP P24387 1/20 0.34
KMT2A Q03164 1/20 0.34
CRHR2 Q13324 1/20 0.34
CTSC P53634 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4420284 0.81 GRN (0.40) CA1CA2PKMKMORAB9A
SCHEMBL14843883 0.81 KMO (0.40) SMN1; SMN2KMOFNTAFNTBPGGT1B
SCHEMBL2800230 0.80 SLC7A5 (0.46) PKMKMO
SCHEMBL4403267 0.78 MDM2 (0.44) SMN1; SMN2KMORAB9ANPC1MEN1
SCHEMBL6897797 0.77 NPC1 (0.38) CA1CA2PKMLMNASMN1; SMN2
SCHEMBL5067808 0.73 HDAC8 (0.41) LMNATSHRRAB9ANPC1ALDH1A1
SCHEMBL2333132 0.71 KMT2A (0.57) LMNASMN1; SMN2TSHRMEN1KMT2A
SCHEMBL7168442 0.71 HSD11B1 (0.42) CA1CA2SMN1; SMN2KMORAB9A
SCHEMBL6228047 0.69 TSHR (0.42) PKMLMNASMN1; SMN2TSHRFNTA
Racemethionine SCHEMBL28833032 0.69 KIF11 (0.48) PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917020-A1 MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS Seattle Genetics, Inc. (US) 2008-05-07 EP disclosed
WO-2007008603-A1 MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS SEATTLE GENETICS, INC. (US) 2007-01-18 WO disclosed