SCHEMBL5069232

SCHEMBL5069232

CC(CC(Cc1cc[c]cc1)c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.43
TAAR1 Q96RJ0 5/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
SIGMAR1 Q99720 2/20 0.38
AOC3 Q16853 2/20 0.37
SLC6A2 P23975 2/20 0.36
MAOA P21397 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CYP2A6 P11509 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
RIPK1 Q13546 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL68592 0.84 ESR1 (0.47) TRPA1TAAR1SIGMAR1AOC3SLC6A2
SCHEMBL27090218 0.81 TRPA1 (0.44) TRPA1TAAR1AOC3SLC6A3RIPK1
SCHEMBL5150293 0.81 ESR1 (0.50) TRPA1TAAR1MTNR1AMTNR1BSIGMAR1
SCHEMBL28163887 0.78 ESR1 (0.53) MTNR1AMTNR1BSIGMAR1AOC3SLC6A2
SCHEMBL3674520 0.78 TRPA1 (0.59) TRPA1TAAR1AOC3SLC6A3RIPK1
SCHEMBL28859481 0.77 ESR1 (0.47) TRPA1TAAR1SIGMAR1SLC6A2MAOA
SCHEMBL7201337 0.77 ESR1 (0.47) TRPA1TAAR1SIGMAR1SLC6A2MAOA
SCHEMBL12816986 0.76 MTNR1A (0.43) TAAR1MTNR1AMTNR1BSIGMAR1SLC6A2
SCHEMBL10437920 0.75 CYP19A1 (0.43) MTNR1AMTNR1B
SCHEMBL4752124 0.74 MTNR1A (0.50) TRPA1TAAR1MTNR1AMTNR1BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7429669-B2 Therapeutic compounds ALLERGAN, INC. (US) 2008-09-30 US disclosed
US-20070293561-A1 5-{3-[(1S,5S)-5-(3-Chloro-5-hydroxymethyl-phenoxymethyl)-4-oxo-cyclopent-2-enyl]-propyl}-thiophene-2-carboxylic acid; Treating eye diseases including glaucoma or ocular hypertension; selective prostaglandin EP2 agonists ALLERGAN, INC. 2007-12-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070293561-A1 5-{3-[(1S,5S)-5-(3-Chloro-5-hydroxymethyl-phenoxymethyl)-4-oxo-cyclopent-2-enyl]-propyl}-thiophene-2-carboxylic acid; Treating eye diseases including glaucoma or ocular hypertension; selective prostaglandin EP2 agonists PTGIR, PTGIS, PTGER2 TRPA1 1818/4885TAAR1 1121/4885MTNR1A 299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.