SCHEMBL5069554

SCHEMBL5069554

Cc1ccc(NC(=O)C(CP(=O)(O)C(Cc2ccccc2)NC(=O)OC(C)(C)C)C(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 10/20 0.48
MME P08473 9/20 0.48
REN P00797 1/20 0.46
HDAC8 Q9BY41 1/20 0.45
MMP8 P22894 1/20 0.43
MMP14 P50281 1/20 0.43
CTSS P25774 2/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSK P43235 1/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KLK5 Q9Y337 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135601 0.90 ECE1 (0.48) ECE1MMEHDAC8MMP8MMP14
SCHEMBL5070528 0.90 ECE1 (0.48) ECE1MMEHDAC8MMP8MMP14
SCHEMBL5071371 0.89 ECE1 (0.55) ECE1MME
SCHEMBL5134614 0.87 ECE1 (0.51) ECE1MMEHDAC8MMP8MMP14
SCHEMBL5041973 0.87 ALDH1A1 (0.49) ECE1MMEHDAC8MMP8MMP14
SCHEMBL5070497 0.78 ECE1 (0.49) ECE1MMERENHDAC8MMP8
SCHEMBL5034289 0.78 ECE1 (0.53) ECE1MMEMMP8MMP14CTSS
SCHEMBL6929264 0.78 ACE2 (0.62) ECE1MME
SCHEMBL5070534 0.77 ECE1 (0.48) ECE1MMEMMP8MMP14CTSS
SCHEMBL5034257 0.76 ECE1 (0.50) ECE1MMECTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685142-B1 PHOSPHINIC ACID DERIVATIVES, BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE HOFFMANN LA ROCHE (CH) 2008-01-09 EP disclosed