SCHEMBL5071371

SCHEMBL5071371

Cc1ccc(NC(=O)C(Cc2ccccc2)CP(=O)(O)C(Cc2ccccc2)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 17/20 0.55
MME P08473 15/20 0.55
ACE2 Q9BYF1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134614 0.94 ECE1 (0.51) ECE1MMEACE2
SCHEMBL5070528 0.90 ECE1 (0.48) ECE1MME
SCHEMBL5135601 0.90 ECE1 (0.48) ECE1MME
SCHEMBL5041973 0.89 ALDH1A1 (0.49) ECE1MME
SCHEMBL5069554 0.89 ECE1 (0.48) ECE1MME
SCHEMBL5070497 0.85 ECE1 (0.49) ECE1MMEACE2
SCHEMBL6929264 0.85 ACE2 (0.62) ECE1MMEACE2
SCHEMBL7621126 0.84 ECE1 (0.74) ECE1MME
SCHEMBL6927137 0.81 ECE1 (0.72) ECE1MME
SCHEMBL5070534 0.79 ECE1 (0.48) ECE1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685142-B1 PHOSPHINIC ACID DERIVATIVES, BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE HOFFMANN LA ROCHE (CH) 2008-01-09 EP disclosed