SCHEMBL5072379

SCHEMBL5072379

O=C(OCCc1cnc(N(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)Cc2cc(C(F)(F)F)cc(Cl)c2OCc2ccccc2)nc1)C1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.43
ALDH1A1 P00352 2/20 0.35
MBTPS1 Q14703 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PIM1 P11309 1/20 0.34
PDGFRA P16234 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
F10 P00742 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL135240 0.86 TACR1 (0.40) TACR1ALDH1A1MEN1KMT2A
SCHEMBL5067467 0.83 TACR1 (0.40) TACR1
SCHEMBL129898 0.82 CETP (0.43) ALDH1A1
SCHEMBL132751 0.78 ALDH1A1 (0.40) TACR1ALDH1A1MEN1KMT2A
SCHEMBL5067463 0.77 TACR1 (0.36) TACR1
SCHEMBL5067462 0.76 TACR1 (0.37) TACR1
SCHEMBL1587634 0.68 SLC6A4 (0.40) TACR1
SCHEMBL130203 0.67 CETP (0.45)
SCHEMBL132026 0.67 CETP (0.45) MEN1KMT2A
SCHEMBL27694957 0.67 AKR1B10 (0.47) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979331-A1 TRISUBSTITUTED AMINE COMPOUNDS AS INHIBITORS OF -CHOLESTERYL ESTER TRANSFER PROTEIN CETP Mitsubishi Tanabe Pharma Corporation (JP) 2008-10-15 EP disclosed
WO-2007088996-A1 TRISUBSTITUTED AMINE COMPOUNDS AS INHIBITORS OF -CHOLESTERYL ESTER TRANSFER PROTEIN CETP MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-08-09 WO disclosed