SCHEMBL5073283

SCHEMBL5073283

COc1ncccc1C(=O)S

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.47
MAPT P10636 3/20 0.46
GAA P10253 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 2/20 0.41
APLNR P35414 1/20 0.41
ALDH1A1 P00352 5/20 0.41
RAB9A P51151 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
NPC1 O15118 2/20 0.41
HTT P42858 1/20 0.41
PPARG P37231 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
BRD4 O60885 1/20 0.41
BRPF1 P55201 1/20 0.41
BTK Q06187 1/20 0.41
SLC13A5 Q86YT5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949562 0.85 TDP1 (0.50) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL18201 0.83 TDP1 (0.57) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL8427582 0.83 TDP1 (0.49) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL30592857 0.83 TDP1 (0.57) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL31081770 0.83 TDP1 (0.49) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL29980732 0.81 RAB9A (0.58) TDP1MAPTGAASMN1; SMN2HPGD
SCHEMBL2488525 0.81 TDP1 (0.47) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL6609846 0.81 TDP1 (0.47) TDP1MAPTGAASMN1; SMN2LMNA
SCHEMBL1723847 0.81 RAB9A (0.58) TDP1MAPTGAASMN1; SMN2HPGD
SCHEMBL311206 0.81 TDP1 (0.69) TDP1MAPTGAASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105246896-B The ketone derivatives of pyrazoles pyrrolizine 4 and its purposes in treatment disease 诺华股份有限公司 2017-09-08 CN disclosed
US-7423168-B2 Reacting allyl starting compound with oxygen nucleophilic agent in presence of transition metal catalyst and monodentate phosphite MITSUBISHI CHEMICAL CORPORATION (JP) 2008-09-09 US disclosed
US-7241857-B2 Method for producing allyl compound, and ether or ester compound produced thereby MITSUBISHI CHEMICAL CORPORATION (JP) 2007-07-10 US disclosed
US-7173157-B2 Method for producing an allyl compound MITSUBISHI CHEMICAL CORPORATION (JP) 2007-02-06 US disclosed
US-7119222-B2 Method for producing allyl compound, and ether or ester compound produced thereby MITSUBISHI CHEMICAL CORPORATION (JP) 2006-10-10 US disclosed
US-20060106181-A1 Method for producing allyl compound, and ether or ester compound produced thereby MITSUBISHI CHEMICAL CORPORATION (JP) 2006-05-18 US disclosed
US-20050075518-A1 Method for producing allyl compound, and allyl compound produced thereby MITSUBISHI CHEMICAL CORPORATION (JP) 2005-04-07 US disclosed
US-20040147757-A1 Method for producing allyl compound, and ether or ester compound produced thereby MITSUBISHI CHEMICAL CORPORATION (JP) 2004-07-29 US disclosed
US-20040092777-A1 Method for producing allyl compound MITSUBISHI CHEMICAL CORPORATION (JP) 2004-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106181-A1 Method for producing allyl compound, and ether or ester compound produced thereby AGPAT5, TST, AGPAT2 TDP1 4654/4885MAPT 2696/4885GAA 2275/4885
US-20040147757-A1 Method for producing allyl compound, and ether or ester compound produced thereby AGPAT5, TST, AGPAT2 TDP1 4654/4885MAPT 2696/4885GAA 2275/4885
US-20040092777-A1 Method for producing allyl compound CCNT1, APEX1, REV1 TDP1 3793/4885MAPT 3604/4885GAA 4745/4885
US-20050075518-A1 Method for producing allyl compound, and allyl compound produced thereby CCNT1, AOC3, ATL3 TDP1 4503/4885MAPT 3247/4885GAA 4076/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.