SCHEMBL5080669

SCHEMBL5080669

CN(C)C(=O)c1cc2c(-c3c(S)nnn3-c3ccc(O)cc3O)cccc2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.34
FLT3 P36888 5/20 0.34
PDGFRB P09619 1/20 0.34
KIT P10721 1/20 0.34
NUDT1 P36639 1/20 0.33
HRH4 Q9H3N8 2/20 0.32
CCNK O75909 1/20 0.32
CDK12 Q9NYV4 1/20 0.32
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973855 0.86 GRIN2D (0.34) HSP90AA1NUDT1HRH4CCNKCDK12
SCHEMBL3978017 0.81 HSP90AA1 (0.34) HSP90AA1
SCHEMBL1343551 0.81 PDK1 (0.35) HSP90AA1PDK1PDK2PDK3PDK4
SCHEMBL3972571 0.81 HSP90AA1 (0.34) HSP90AA1
SCHEMBL1147866 0.77 HSD11B1 (0.32) HSP90AA1
SCHEMBL1147785 0.77 PIK3CD (0.36) HSP90AA1
SCHEMBL3971042 0.76 HSP90AA1 (0.32) HSP90AA1
SCHEMBL930756 0.75 ESR1 (0.39) HSP90AA1
SCHEMBL1148407 0.75 GAA (0.36) HSP90AA1
SCHEMBL1502369 0.74 FLT3 (0.37) HSP90AA1FLT3PDGFRBKITNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051416-A2 COMPOUNDS THAT INHIBIT THE ACTIVITY OF HSP90 FOR TREATING INFECTIONS SYNTA PHARMACEUTICALS CORP. (US) 2008-05-02 WO disclosed