SCHEMBL5083213

SCHEMBL5083213

COCCOc1ccccc1-c1ccccc1-c1[c]nns1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.42
ADRB2 P07550 2/20 0.39
HTR7 P34969 2/20 0.38
AR P10275 2/20 0.36
KDM4E B2RXH2 4/20 0.35
PDE5A O76074 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLQ O75417 1/20 0.33
IDO1 P14902 1/20 0.33
ADRB1 P08588 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5081008 0.93 KDM4E (0.40) KCNN4ADRB2HTR7KDM4EL3MBTL1
SCHEMBL5083181 0.86 KDM4E (0.41) KCNN4ADRB2HTR7KDM4EPDE5A
SCHEMBL5083191 0.86 KDM4E (0.41) KCNN4ADRB2HTR7KDM4EPDE5A
SCHEMBL5087245 0.83 CYP1A2 (0.35) ADRB2HTR7KDM4EPDE5AL3MBTL1
SCHEMBL4721568 0.82 PDE5A (0.41) ADRB2KDM4EPDE5AALDH1A1LMNA
SCHEMBL4723651 0.81 CYP1A2 (0.48) KDM4EPDE5ACYP1A2CYP2C19
SCHEMBL4723561 0.79 ALDH1A1 (0.40) KDM4EPDE5AALDH1A1MEN1KMT2A
SCHEMBL5083208 0.78 KCNN4 (0.31) KCNN4KDM4EALDH1A1TSHR
SCHEMBL478309 0.77 HTR7 (0.56) KCNN4ADRB2HTR7ARKDM4E
SCHEMBL4724808 0.76 APP (0.46) KDM4EL3MBTL1ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7375081-B2 Therapeutic combination of a pneumocandin derivative and an antifungal agent ASTELLAS PHARMA INC. (JP) 2008-05-20 US claimed
US-6875740-B1 Combination of a cyclic hexapeptide with antifungal drugs for treatment of fungal pathogens FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2005-04-05 US claimed