SCHEMBL5087799

SCHEMBL5087799

Nc1cc2ccccc2n1C1CC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.44
OPRD1 P41143 10/20 0.44
OPRK1 P41145 10/20 0.44
OPRL1 P41146 9/20 0.44
RPS6KB1 P23443 4/20 0.43
ROCK1 Q13464 4/20 0.43
PRKACA P17612 3/20 0.38
GSK3B P49841 3/20 0.38
OGFRL1 Q5TC84 1/20 0.38
CYP11B2 P19099 2/20 0.36
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30995223 0.93 ROCK1 (0.46) OPRM1OPRD1OPRK1OPRL1RPS6KB1
SCHEMBL16103839 0.77 OPRM1 (0.44) OPRM1OPRD1OPRK1OPRL1CYP11B2
SCHEMBL30995117 0.76 CYP11B2 (0.44) CYP11B2CYP11B1
SCHEMBL30344944 0.74 KMT2A (0.53) OPRM1OPRD1OPRK1OPRL1CYP11B2
SCHEMBL30995183 0.74 PRKACA (0.37) RPS6KB1ROCK1PRKACAGSK3B
SCHEMBL30995162 0.74 CYP11B2 (0.44) OPRM1OPRL1RPS6KB1ROCK1PRKACA
SCHEMBL28330578 0.74 PLA2G10 (0.47) OPRM1OPRD1OPRK1OPRL1OGFRL1
SCHEMBL30995229 0.73 ABL1 (0.37) OPRM1CYP11B2CYP11B1
SCHEMBL12491808 0.73 OPRM1 (0.41) OPRM1OPRD1OPRK1OPRL1OGFRL1
SCHEMBL12490206 0.73 OPRM1 (0.67) OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007756-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmceuticals Incorporated (US) 2008-12-31 EP disclosed
WO-2007117715-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-18 WO disclosed