SCHEMBL5088070

SCHEMBL5088070

CCOC(=O)c1c(C)nc(Nc2cccc(Cl)c2)c2nc[nH]c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
MAPT P10636 4/20 0.52
KDM4E B2RXH2 3/20 0.52
BRAF P15056 2/20 0.52
ALOX5 P09917 2/20 0.49
PTGES O14684 1/20 0.49
HPGD P15428 2/20 0.44
TRPV1 Q8NER1 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 2/20 0.42
TP53 P04637 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPK1 P28482 1/20 0.41
EGFR P00533 1/20 0.41
SIRT5 Q9NXA8 1/20 0.41
MEN1 O00255 1/20 0.41
CSNK2A2 P19784 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5087476 0.87 EGFR (0.49) BRAFKMT2AEGFRMEN1CSNK2A2
SCHEMBL5087486 0.76 KDM4E (0.43) ALDH1A1MAPTKDM4EHPGDNPC1
SCHEMBL10488563 0.75 SMN1; SMN2 (0.56) ALDH1A1MAPTKDM4EALOX5PTGES
SCHEMBL4898607 0.74 BRAF (0.61) ALDH1A1MAPTKDM4EBRAFHPGD
SCHEMBL3993488 0.71 MAPT (0.55) ALDH1A1MAPTKDM4EALOX5PTGES
SCHEMBL28426697 0.70 MEN1 (0.60) ALDH1A1MAPTKDM4EALOX5PTGES
SCHEMBL16146826 0.70 BRAF (0.51) BRAFKMT2AEGFRMEN1CSNK2A2
SCHEMBL9896825 0.70 JAK3 (0.68) EGFRJAK2JAK3
Hydrochloric Acid SCHEMBL9896822 0.69 JAK3 (0.67) EGFRJAK2JAK3
SCHEMBL5250340 0.69 TTBK1 (0.48) ALDH1A1KMT2AEGFRMEN1CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008116816-A1 COMBINATION OF CB2 LIGAND AND PARACETAMOL GLAXO GROUP LIMITED (GB) 2008-10-02 WO disclosed