SCHEMBL5120128

SCHEMBL5120128

CC(C)C1CC(c2nc(O)c(O)c(C(=O)NCc3ccc(F)cc3)n2)N(C)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
POLB P06746 1/20 0.43
KCNE1 P15382 1/20 0.42
CCR1 P32246 1/20 0.42
KCNQ1 P51787 1/20 0.42
KCNH2 Q12809 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALDH1A1 P00352 4/20 0.40
HTT P42858 1/20 0.40
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ERCC1 P07992 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
HMGCR P04035 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5121129 0.87 KCNE1 (0.44) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2
SCHEMBL5129303 0.83 SMN1; SMN2 (0.43) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2
SCHEMBL5122833 0.82 SMN1; SMN2 (0.40) SMN1; SMN2POLBKCNE1CCR1KCNQ1
SCHEMBL5119559 0.82 KCNE1 (0.44) SMN1; SMN2POLBKCNE1CCR1KCNQ1
SCHEMBL5116540 0.82 KCNE1 (0.45) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2
SCHEMBL5128153 0.82 KCNE1 (0.46) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2
SCHEMBL5114548 0.81 CALCA (0.42) SMN1; SMN2POLBKCNE1CCR1KCNQ1
SCHEMBL5123596 0.81 LMNA (0.43) SMN1; SMN2KCNE1CCR1KCNQ1ALDH1A1
SCHEMBL5128477 0.81 KCNH2 (0.50) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2
SCHEMBL5115008 0.80 KCNE1 (0.44) SMN1; SMN2KCNE1CCR1KCNQ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459452-B2 Dihydroxypyrimidine carboxamide inhibitors of HIV integrase ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2008-12-02 US claimed