SCHEMBL5127724

SCHEMBL5127724

CNC(=O)c1ccc(-c2ccc3nc(N)nc(OCCF)c3c2)cc1.Nc1nc(OC[C@@H]2CCCO2)c2cc(-c3ccc(C(=O)NC4CC4)cc3)ccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.45
NPC1 O15118 6/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
MAPK14 Q16539 2/20 0.42
CYP2C9 P11712 1/20 0.42
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 3/20 0.40
HPGD P15428 2/20 0.40
MAPK1 P28482 1/20 0.40
PTK2 Q05397 2/20 0.40
TP53 P04637 2/20 0.40
RIPK2 O43353 1/20 0.40
AXL P30530 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340899 0.91 RAB9A (0.53) RAB9ANPC1SMN1; SMN2MAPK14CYP2C9
SCHEMBL3340903 0.91 RAB9A (0.53) RAB9ANPC1SMN1; SMN2MAPK14CYP2C9
SCHEMBL3335167 0.86 SMYD3 (0.47) RAB9ANPC1SMN1; SMN2MAPK14CYP2C9
SCHEMBL3334272 0.84 SMYD3 (0.43) RAB9ANPC1SMN1; SMN2MAPK14MEN1
SCHEMBL3334266 0.82 PIK3CA (0.42) ALDH1A1MCHR1
SCHEMBL3332984 0.81 MEN1 (0.46) RAB9ANPC1SMN1; SMN2MAPK14CYP2C9
SCHEMBL3337490 0.79 LMNA (0.44) RAB9ANPC1SMN1; SMN2MAPK14MEN1
SCHEMBL3334542 0.78 MEN1 (0.45) RAB9ANPC1SMN1; SMN2MAPK14CYP2C9
SCHEMBL5129389 0.78 BMPR1B (0.43) MAPK14ALDH1A1LMNAHPGDTP53
SCHEMBL3336243 0.78 TRIM58 (0.48) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed