SCHEMBL5132644

SCHEMBL5132644

CC(C)(C)CC(=O)c1cc2cc([N+](=O)[O-])cc(C(=O)O)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 2/20 0.40
APEX1 P27695 1/20 0.38
HTT P42858 2/20 0.37
TP53 P04637 1/20 0.37
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
AKR1B1 P15121 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1465571 0.78 ALDH1A1 (0.40) HTTTP53ALDH1A1MAPTAKR1B1
SCHEMBL12501374 0.71 APEX1 (0.51) FBP1APEX1ALDH1A1KMT2ACYP1A2
SCHEMBL30856079 0.70 MAOA (0.45) APEX1HTTTP53ALDH1A1MAPT
SCHEMBL12501380 0.68 APEX1 (0.51) FBP1APEX1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL12501291 0.68 ALDH1A1 (0.56) FBP1APEX1HTTALDH1A1MAPT
SCHEMBL2919368 0.67 MAPT (0.42) HTTTP53ALDH1A1MAPTAKR1B1
SCHEMBL11420063 0.66 ALDH1A1 (0.49) HTTTP53ALDH1A1MAPTKMT2A
SCHEMBL13956351 0.65 L3MBTL1 (0.61) HTTTP53ALDH1A1MAPTKMT2A
SCHEMBL14651329 0.65 KMT2A (0.47) FBP1APEX1HTTALDH1A1KMT2A
SCHEMBL1466537 0.65 XDH (0.41) HTTALDH1A1MAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007756-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmceuticals Incorporated (US) 2008-12-31 EP disclosed
WO-2007117715-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-18 WO disclosed