Bromide

Bromide

SCHEMBL5133339

CCOC(=O)CCCN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)OC(C)(C)C)CC1.[Br-].[Na+]

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH2 known ✓ P25021 1/20 0.32
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 2/20 0.35
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SIGMAR1 Q99720 3/20 0.33
HTR4 Q13639 1/20 0.33
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
FKBP1A P62942 1/20 0.32
TNF P01375 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
HRH1 P35367 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL5125778 0.96 RAB9A (0.34) RAB9AL3MBTL1CYP1A2SIGMAR1PTGDR2
Bromide SCHEMBL5133338 0.89 RAB9A (0.34) RAB9AL3MBTL1CYP1A2SIGMAR1HTR4
SCHEMBL16656257 0.88 RAB9A (0.36) RAB9AL3MBTL1CYP1A2SIGMAR1HTR4
Bromide SCHEMBL5125776 0.86 L3MBTL1 (0.34) RAB9AL3MBTL1CYP1A2HTR4LMNA
Bromide SCHEMBL5132382 0.86 CYP1A2 (0.47) CYP1A2MAPK1SMN1; SMN2SIGMAR1
Bromide SCHEMBL5126215 0.83 PLA2G10 (0.34) SMN1; SMN2SIGMAR1TSHRKDM4E
Bromide SCHEMBL5133205 0.82 CYP1A2 (0.42) CYP1A2MAPK1SMN1; SMN2SIGMAR1
SCHEMBL18748496 0.80 LMNA (0.35) SMN1; SMN2SIGMAR1LMNAPOLBTSHR
SCHEMBL20678139 0.80 HSD17B10 (0.36) SMN1; SMN2SIGMAR1TSHRKDM4E
SCHEMBL17119745 0.80 HSD17B10 (0.36) SMN1; SMN2SIGMAR1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134289-A2 HIGH RELAXIVITY COORDINATIVELY UNSATURATED LANTHANIDE COMPLEXES MALLINCKRODT INC. (US) 2008-11-06 WO disclosed