SCHEMBL5133752

SCHEMBL5133752

CCCc1nn(C)c2cnc(N(C)c3ccnc(N4CCOCC4)c3)nc12

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.39
LRRK2 Q5S007 9/20 0.37
PIK3CA P42336 2/20 0.36
ATR Q13535 6/20 0.35
ATRIP Q8WXE1 5/20 0.35
CSF1R P07333 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133754 0.78 OGA (0.40) LRRK2PIK3CA
SCHEMBL4903928 0.77 PDE5A (0.46) KDM4CHDAC1
SCHEMBL5134689 0.70 RORC (0.35) HDAC1
SCHEMBL13069962 0.66 PIK3CA (0.53) LRRK2PIK3CA
SCHEMBL4903908 0.64 PDE5A (0.45) PIK3CAHDAC1
SCHEMBL5134146 0.62 LMNA (0.38) HDAC1
SCHEMBL3122462 0.62 PDE5A (0.36)
SCHEMBL18765799 0.61 PIK3CA (0.57) KDM4CLRRK2PIK3CA
SCHEMBL14554006 0.61 SORD (0.51) PIK3CA
SCHEMBL17916959 0.61 LRRK2 (0.46) LRRK2PIK3CAATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO claimed
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO disclosed