SCHEMBL5134656

SCHEMBL5134656

COCCOC1=C(C)C(=O)C(c2ncnc3ccccc23)=C(N)C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.42
ADORA2A P29274 1/20 0.38
TSHR P16473 3/20 0.37
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.36
KDM1A O60341 4/20 0.36
MPO P05164 1/20 0.36
FFAR2 O15552 1/20 0.34
KIT P10721 1/20 0.33
NCF1 P14598 2/20 0.33
EGFR P00533 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5664809 0.83 LDHA (0.40) LDHAADORA2ATSHRPI4KAPI4K2B
SCHEMBL5135024 0.74 ADORA2A (0.43) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL5135022 0.72 ADORA2A (0.44) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL5134655 0.70 TLR7 (0.38) TSHRL3MBTL1MPONCF1ALDH1A1
SCHEMBL5665202 0.68 KDR (0.42) KDM1AKITEGFR
SCHEMBL5134739 0.67 MAP4K4 (0.40) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL5135030 0.67 GAPDH (0.42) ADORA2ATSHRPI4KAPI4K2BPI4K2A
SCHEMBL5664802 0.67 TLR7 (0.40) ADORA2ATSHRL3MBTL1KDM1AMPO
SCHEMBL5664940 0.66 KDR (0.43) KDM1AKITEGFR
SCHEMBL5135370 0.66 CES1 (0.47) ADORA2ARAB9ANPC1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080268460-A1 Assays to Identify Irreversibly Binding Inhibitors of Receptor Tyrosine Kinases WYETH (US) 2008-10-30 US disclosed