SCHEMBL5136650

SCHEMBL5136650

CCOC(=O)n1c(C(=O)Cl)cc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 6/20 0.55
NOD1 Q9Y239 6/20 0.55
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
KDM4E B2RXH2 1/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
F10 P00742 1/20 0.46
GAA P10253 3/20 0.45
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CYP2D6 P10635 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988991 0.87 NOD2 (0.71) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL3972260 0.81 NOD2 (0.53) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL4251782 0.81 NR1H2 (0.54)
SCHEMBL29725642 0.81 NR1H2 (0.54)
SCHEMBL27570092 0.79 DAO (0.49) NOD2NOD1MAPTCYP1A2MCL1
SCHEMBL8689345 0.79 KMT2A (0.58) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL28615205 0.79 NOD2 (0.51) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL6706688 0.79 NOD2 (0.51) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL4056238 0.78 NOD2 (0.50) NOD2NOD1MEN1KMT2ASMN1; SMN2
SCHEMBL24894603 0.77 NOD2 (0.62) NOD2NOD1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904477-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed