SCHEMBL4056238

SCHEMBL4056238

CCOC(=O)n1c(OC)cc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 3/20 0.50
NOD1 Q9Y239 3/20 0.50
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
GAA P10253 3/20 0.44
PSMD14 O00487 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
ALDH1A1 P00352 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
NR1H2 P55055 1/20 0.42
LMNA P02545 2/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.41
GLA P06280 1/20 0.41
NTRK1 P04629 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11980494 0.85 NOD2 (0.48) NOD2NOD1MEN1KMT2AGAA
SCHEMBL3972260 0.83 NOD2 (0.53) NOD2NOD1MEN1KMT2AGAA
SCHEMBL3847463 0.81 MCL1 (0.45) NOD2NOD1MEN1KMT2AALDH1A1
SCHEMBL28370896 0.81 NR1H2 (0.55) NR1H2
SCHEMBL28615205 0.80 NOD2 (0.51) NOD2NOD1MEN1KMT2AGAA
SCHEMBL6706688 0.80 NOD2 (0.51) NOD2NOD1MEN1KMT2AGAA
SCHEMBL11890112 0.79 NR1H2 (0.43) NOD2NOD1MEN1KMT2AGAA
SCHEMBL6988991 0.79 NOD2 (0.71) NOD2NOD1MEN1KMT2AGAA
SCHEMBL28455040 0.78 NOD2 (0.47) NOD2NOD1MEN1KMT2AGAA
SCHEMBL5136650 0.78 NOD2 (0.55) NOD2NOD1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009097515-A2 [A]-FUSED INDOLE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-08-06 WO disclosed
EP-1966134-A1 NOVEL FUSED PYRROLE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-09-10 EP disclosed
WO-2007068621-A1 NOVEL FUSED PYRROLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-06-21 WO disclosed