SCHEMBL5137969

SCHEMBL5137969

Cc1cccc2c1Cc1ccccc1C(=O)N2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.53
CASP6 P55212 2/20 0.53
TDP2 O95551 1/20 0.53
CASP7 P55210 1/20 0.53
CASP9 P55211 1/20 0.53
CASP8 Q14790 1/20 0.53
MAP3K14 Q99558 1/20 0.53
POLB P06746 1/20 0.47
ACVR1 Q04771 2/20 0.44
LRRK2 Q5S007 2/20 0.44
PDGFRA P16234 1/20 0.44
FER P16591 1/20 0.44
LTK P29376 1/20 0.44
CDK8 P49336 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
PARP1 P09874 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP11 Q9NR21 1/20 0.44
CDK5 Q00535 2/20 0.43
CCNB2 O95067 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852644 0.81 CASP7 (0.53) CASP3CASP6TDP2CASP7CASP9
SCHEMBL5141694 0.80 NPC1 (0.47) CDK5CCNB2CDK1CCNB1GSK3B
SCHEMBL2087698 0.78 TDP2 (0.66) CASP3CASP6TDP2CASP7CASP9
SCHEMBL14084317 0.75 TDP2 (0.61) CASP3CASP6TDP2CASP7CASP9
SCHEMBL10694265 0.75 MAOA (0.61) CASP3CASP6PARP1PARP10PARP11
SCHEMBL29622074 0.74 CCNB2 (0.54) CDK5CCNB2CDK1CCNB1GSK3B
SCHEMBL152281 0.74 CCNB2 (0.54) CDK5CCNB2CDK1CCNB1GSK3B
SCHEMBL135721 0.74 PNMT (0.53) CASP3CASP6PARP1PARP10PARP11
SCHEMBL27878508 0.74 PNMT (0.53) CASP3CASP6PARP1PARP10PARP11
SCHEMBL12834903 0.74 AHR (0.53) TDP2POLBLRRK2PARP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924580-A1 NON-STEROIDAL COMPOUNDS USEFUL AS GLUCOCORTICOID RECEPTOR MODULATORS N.V. Organon (NL) 2008-05-28 EP disclosed
WO-2007025938-A1 NON-STEROIDAL COMPOUNDS USEFUL AS GLUCOCORTICOID RECEPTOR MODULATORS N.V. ORGANON (NL) 2007-03-08 WO disclosed