SCHEMBL51386

SCHEMBL51386

CN1C(C)(C)CN(c2cc(F)ccc2CN)S1(O)O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AMPD2 Q01433 3/20 0.38
NCF1 P14598 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
MPO P05164 1/20 0.31
TRPA1 O75762 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL52723 0.99 AMPD2 (0.37) AMPD2NCF1ALDH1A1L3MBTL1HDAC1
SCHEMBL51385 0.85 AMPD2 (0.37) AMPD2NCF1ALDH1A1L3MBTL1MPO
SCHEMBL52326 0.76 FFAR4 (0.38) AMPD2HDAC1HDAC6
SCHEMBL12215851 0.71 CRY1 (0.39) NCF1ALDH1A1L3MBTL1P2RX7
SCHEMBL29817889 0.71 ALDH1A1 (0.59) NCF1ALDH1A1L3MBTL1MPO
Hydrochloric Acid SCHEMBL2528915 0.70 CRY1 (0.39) NCF1ALDH1A1L3MBTL1P2RX7
SCHEMBL12215772 0.66 CA1 (0.40)
Hydrochloric Acid SCHEMBL2531492 0.65 CA1 (0.39) ALDH1A1
SCHEMBL52688 0.65 P2RX7 (0.41) ALDH1A1L3MBTL1P2RX7
Hydrochloric Acid SCHEMBL2531529 0.64 P2RX7 (0.40) ALDH1A1L3MBTL1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280981-B1 BRIDGED HETEROCYCLES AS HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-04-23 EP disclosed
US-8129398-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-06 US disclosed
US-20090253677-A1 HIV Integrase Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090253677-A1 HIV Integrase Inhibitors DNTT, POLB, UNG AMPD2 797/4885NCF1 1037/4885ALDH1A1 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.