SCHEMBL5138939

SCHEMBL5138939

c1cncc(-c2ccc[nH]2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 7/20 0.60
CYP3A4 P08684 3/20 0.60
CYP2E1 P05181 2/20 0.60
CYP2B6 P20813 2/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
BCHE P06276 1/20 0.51
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP19A1 P11511 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29422979 1.00 CYP2A6 (0.60) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
Pyrazole SCHEMBL28013454 0.88 CYP2A6 (0.49) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
SCHEMBL162771 0.80
Pyridine SCHEMBL28139351 0.79 CYP3A4 (0.45) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
Hydrochloric Acid SCHEMBL6647002 0.78 CYP2A6 (0.53) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
Hydrochloric Acid SCHEMBL28088469 0.78 CYP2A6 (0.53) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
SCHEMBL8013084 0.78 ATM (0.44) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
Pyridine SCHEMBL28547162 0.78 CYP3A4 (0.44) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
SCHEMBL29827246 0.77 CYP2A6 (0.53) CYP2A6CYP3A4CYP2E1CYP2B6CYP2D6
SCHEMBL2457937 0.77 CHRNB2 (0.67) ALDH1A1KDM4ETP53MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11939291-B2 GRP94 selective inhibitors and uses thereof UNIVERSITY OF KANSAS (US) 2024-03-26 US disclosed
US-20230391752-A1 PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AND RELATED USES CHULALONGKORN UNIVERSITY (TH) 2023-12-07 US disclosed
CN-110452243-B Pyrrolopyrimidine derivative epidermal growth factor inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2022-11-11 CN disclosed
CN-114746090-A Azaindole carboxamide compounds for the treatment of mycobacterial infections 结核病药物开发全球联盟公司 2022-07-12 CN disclosed
US-20220024869-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF UNIVERSITY OF KANSAS 2022-01-27 US disclosed
US-20220024869-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF UNIVERSITY OF KANSAS 2022-01-27 US disclosed
US-20220008891-A1 PROCESS FOR CONDITIONING METAL-ORGANIC FRAMEWORKS BY MEANS OF MEMBRANE FILTRATION BASF SE (DE) 2022-01-13 US disclosed
US-20210289832-A1 LIPOPHILIC ACTIVE AGENT INFUSED TOBACCO LEAVES AND/OR TOBACCO MATERIALS AND METHODS OF USE THEREOF Poviva Corp. (US) 2021-09-23 US disclosed
US-20210213091-A1 LIPOPHILIC ACTIVE AGENT INFUSED TOBACCO LEAVES AND/OR TOBACCO MATERIALS AND METHODS OF USE THEREOF Poviva Corp. (US) 2021-07-15 US disclosed
US-20210145818-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF Poviva Corp. 2021-05-20 US disclosed
CN-101175747-A Substituted N-arylpyrrolidines as selective androgen receptor modulators LILLY CO ELI (US) 2008-05-07 CN disclosed
US-20070072001-A1 Luminescent device CANON KABUSHIKI KAISHA (JP) 2007-03-29 US disclosed
US-20070072001-A1 Luminescent device CANON KABUSHIKI KAISHA (JP) 2007-03-29 US disclosed
US-20040198730-A1 Pyridylfurans and pyrroles as raf kinase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2004-10-07 US disclosed
EP-1432699-A1 PYRIDYLFURANS AND PYRROLES AS RAF KINASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2004-06-30 EP disclosed
WO-2003027101-A1 SUBSTITUTED 3-PYRIDYL PYRROLES AND 3-PYRIDYL PYRAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed
WO-2003027101-A1 SUBSTITUTED 3-PYRIDYL PYRROLES AND 3-PYRIDYL PYRAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed
WO-2003022832-A1 PYRIDYLFURANS AND PYRROLES AS RAF KINASE INHIBITORS SMITHKLINE BEECHAM P.L.C. (GB) 2003-03-20 WO disclosed
EP-0103969-B1 PRINTING INKS AND PRINTED SUBSTRATES LAWRENCE, Peter Robin Broughton (GB) 1986-10-29 EP disclosed
US-4574151-A Amine salts and products containing them Lawrence, Peter Robin Broughton (GB) 1986-03-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040198730-A1 Pyridylfurans and pyrroles as raf kinase inhibitors BRAF, ARAF, RAF1 CYP2A6 3714/4885CYP3A4 3513/4885CYP2E1 2713/4885
US-20230391752-A1 PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AND RELATED USES GLS2, PYGL, CPS1 CYP2A6 160/4885CYP3A4 34/4885CYP2E1 5/4885
US-20210145818-A1 COMPOSITIONS INFUSED WITH NICOTINE COMPOUNDS AND METHODS OF USE THEREOF CHRNA5, SLC18A3, CHRNA6 CYP2A6 1222/4885CYP3A4 1962/4885CYP2E1 2509/4885
US-11939291-B2 GRP94 selective inhibitors and uses thereof GRPR, HSP90B1, HSPE1 CYP2A6 4220/4885CYP3A4 3988/4885CYP2E1 4348/4885
US-20220024869-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF GRPR, HSP90B1, HSPE1 CYP2A6 4220/4885CYP3A4 3988/4885CYP2E1 4348/4885
US-20220008891-A1 PROCESS FOR CONDITIONING METAL-ORGANIC FRAMEWORKS BY MEANS OF MEMBRANE FILTRATION CD69, OSTC, OGFR CYP2A6 2798/4885CYP3A4 2853/4885CYP2E1 2183/4885
US-20210213091-A1 LIPOPHILIC ACTIVE AGENT INFUSED TOBACCO LEAVES AND/OR TOBACCO MATERIALS AND METHODS OF USE THEREOF MGLL, LIPA, LAMP1 CYP2A6 2861/4885CYP3A4 2893/4885CYP2E1 3766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.