SCHEMBL5139150

SCHEMBL5139150

O=C(NC1=CCCCC1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
TP53 P04637 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
GAA P10253 2/20 0.46
NFKB1 P19838 1/20 0.46
HTT P42858 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
PTPN1 P18031 2/20 0.44
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 2/20 0.43
SIRT1 Q96EB6 1/20 0.43
KDM4E B2RXH2 1/20 0.43
FLT3 P36888 1/20 0.43
HDAC3 O15379 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10427470 0.95 NPC1 (0.47) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL5585822 0.78 NPC1 (0.51) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL12336002 0.78 PTGS2 (0.53) NPC1RAB9ASMN1; SMN2GAAMEN1
SCHEMBL5932198 0.77 HDAC2 (0.44) NPC1RAB9ASMN1; SMN2HTTALDH1A1
SCHEMBL27797782 0.76 RAB9A (0.57) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL5932189 0.74 HDAC2 (0.44) NPC1RAB9ASMN1; SMN2NFKB1HTT
SCHEMBL12757508 0.72 SERPINE1 (0.52) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL14099881 0.72 NPC1 (0.50) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL25095364 0.72 HDAC2 (0.42) NPC1RAB9ASMN1; SMN2NFKB1HTT
SCHEMBL5932684 0.72 HDAC2 (0.42) NPC1RAB9ASMN1; SMN2NFKB1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7326700-B2 Cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists WYETH (US) 2008-02-05 US disclosed
US-6903087-B2 For prevention and/or suppression of preterm labor, suppression of labor at term prior to caesarean delivery, and for the treatment of dysmenorrhea; useful in enhancing fertility rates WYETH (US) 2005-06-07 US disclosed
US-20030055046-A1 Novel pyrido cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists WYETH 2003-03-20 US disclosed
US-20030004159-A1 Novel cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists WYETH 2003-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030055046-A1 Novel pyrido cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists OXTR, OPRL1, PRLHR NPC1 4637/4885RAB9A 4783/4885TP53 4728/4885
US-20030004159-A1 Novel cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists OXTR, OPRL1, HCRTR2 NPC1 4166/4885RAB9A 4755/4885TP53 4770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.