SCHEMBL5139850

SCHEMBL5139850

CC(N)(c1ccccc1)c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.40
MTOR P42345 1/20 0.40
ADK P55263 1/20 0.40
NISCH Q9Y2I1 1/20 0.40
TAAR1 Q96RJ0 7/20 0.37
KDM4E B2RXH2 1/20 0.36
KCNN4 O15554 1/20 0.35
SLC6A2 P23975 1/20 0.34
CDC7 O00311 1/20 0.34
MAP4K4 O95819 1/20 0.34
PIM1 P11309 1/20 0.34
PRKACA P17612 1/20 0.34
GSK3B P49841 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7838270 0.82 ALDH1A1 (0.42) CYP19A1MTORADKNISCHALDH1A1
SCHEMBL2697752 0.81 MTOR (0.42) CYP19A1MTORADKNISCHTAAR1
SCHEMBL6302051 0.79 CYP19A1 (0.47) CYP19A1MTORADKNISCHTAAR1
SCHEMBL697087 0.79 CYP19A1 (0.47) CYP19A1MTORADKNISCHTAAR1
SCHEMBL5240030 0.78 CYP1A2 (0.38) CYP19A1MTORADKNISCHTAAR1
SCHEMBL11089506 0.77 MTOR (0.45) CYP19A1MTORADKNISCHTAAR1
Trityl Imidazole SCHEMBL1572623 0.77 MTOR (0.45) CYP19A1MTORADKNISCHTAAR1
SCHEMBL5380824 0.74
SCHEMBL6090949 0.74 CYP19A1 (0.64) CYP19A1MTORADKNISCHTAAR1
SCHEMBL5676876 0.74 CYP19A1 (0.46) CYP19A1MTORADKNISCHTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7326792-B2 Heterocyclic compounds as P2X7 ion channel blockers AVENTIS PHARMACEUTICALS INC. (US) 2008-02-05 US disclosed
US-20050026916-A1 Heterocyclic compounds as P2X7 ion channel blockers AVENTIS PHARMACEUTICALS INC. (US) 2005-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050026916-A1 Heterocyclic compounds as P2X7 ion channel blockers P2RX3, P2RX2, P2RX5 CYP19A1 3562/4885MTOR 2926/4885ADK 479/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.