SCHEMBL5140428

SCHEMBL5140428

Cc1c(C(F)(F)F)c(C(N)=O)cc(C2CCN(CC3CCOCC3)CC2)c1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.39
EBP Q15125 5/20 0.38
BRD4 O60885 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
OPRM1 P35372 2/20 0.35
PARP1 P09874 1/20 0.35
NAMPT P43490 1/20 0.35
KCNH2 Q12809 1/20 0.35
RBP4 P02753 1/20 0.35
LMNA P02545 1/20 0.34
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135453 0.83 THRB (0.40) THRBBRD4OPRM1PARP1NAMPT
SCHEMBL5134528 0.82 THRB (0.38) THRBBRD4CNR1CNR2OPRM1
SCHEMBL5140672 0.81 PARP2 (0.40) PARP1KCNH2
SCHEMBL5146830 0.79 ALDH1A1 (0.40) OPRM1PARP1KCNH2
SCHEMBL5190872 0.78 PARP1 (0.42) THRBBRD4OPRM1PARP1NAMPT
SCHEMBL5136171 0.72 PARP1 (0.45) CNR1CNR2PARP1NAMPTKCNH2
SCHEMBL5531782 0.68 KDM4E (0.42) PARP1KCNH2
SCHEMBL5527850 0.66 KDM4E (0.42) PARP1KCNH2
SCHEMBL5136169 0.65 NAMPT (0.41) CNR1CNR2OPRM1PARP1NAMPT
SCHEMBL1438737 0.64 SMN1; SMN2 (0.53) THRBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed