SCHEMBL5140765

SCHEMBL5140765

Cc1cccc(C)c1NC(=O)[AsH]c1ccc(-c2ccc(C(=O)N3CCC[C@@H]3C(=O)O)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
ITGB3 P05106 1/20 0.48
ITGB1 P05556 1/20 0.48
ITGAV P06756 1/20 0.48
ITGA5 P08648 1/20 0.48
ITGA4 P13612 1/20 0.48
ALDH1A1 P00352 3/20 0.47
CA2 P00918 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
DGAT1 O75907 7/20 0.46
HPGD P15428 1/20 0.45
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3094864 0.87 DGAT1 (0.58) NPSR1ITGB3ITGB1ITGAVITGA5
SCHEMBL3092210 0.84 DGAT1 (0.55) NPSR1ITGB3ITGB1ITGAVITGA5
SCHEMBL5140198 0.82 TDP1 (0.47) NPSR1ITGB3ITGB1ITGAVITGA5
SCHEMBL3103290 0.78 DGAT1 (0.56) ITGB3ITGB1ITGAVITGA5ITGA4
SCHEMBL5036076 0.77 CA2 (0.64) NPSR1ALDH1A1CA2L3MBTL1DGAT1
SCHEMBL1750558 0.77 CA2 (0.64) NPSR1ALDH1A1CA2L3MBTL1DGAT1
SCHEMBL24313493 0.77 ALDH1A1 (0.56) NPSR1ITGB3ITGB1ITGAVITGA5
SCHEMBL3105657 0.75 DGAT1 (0.53) ITGB3ITGB1ITGAVITGA5ITGA4
SCHEMBL3103397 0.75 DGAT1 (0.57) NPSR1ALDH1A1CA2L3MBTL1DGAT1
SCHEMBL5537767 0.74 CA2 (0.75) NPSR1ALDH1A1CA2L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912634-A2 PREPARATION AND USE OF BIPHENYL AMINO ACID DERIVATIVES FOR THE TREATMENT OF OBESITY Bayer Healthcare, LLC (US) 2008-04-23 EP claimed
WO-2007016538-A2 PREPARATION AND USE OF BIPHENYL AMINO ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2007-02-08 WO claimed