SCHEMBL5141689

SCHEMBL5141689

CN(C)C(=O)N(c1ccccc1)c1cc[nH]n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.46
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGIR P43119 1/20 0.36
KMT2A Q03164 4/20 0.36
TSHR P16473 3/20 0.36
HTT P42858 3/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GLA P06280 1/20 0.36
CHRM4 P08173 3/20 0.36
CHRM3 P20309 3/20 0.36
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
CHRM2 P08172 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400582 0.89 NPSR1 (0.44) NPSR1ATMTDP1L3MBTL1PTGIR
SCHEMBL6905225 0.83 KMT2A (0.46) NPSR1ATMTDP1L3MBTL1KMT2A
SCHEMBL4458935 0.83 NPSR1 (0.47) NPSR1ATMTDP1L3MBTL1KMT2A
SCHEMBL398536 0.80 NPSR1 (0.44) NPSR1ATMTDP1L3MBTL1PTGIR
SCHEMBL3424139 0.79 SMN1; SMN2 (0.44) NPSR1ATMTDP1L3MBTL1KMT2A
SCHEMBL748812 0.78 NPSR1 (0.73) NPSR1ATMTDP1L3MBTL1PTGIR
SCHEMBL27960846 0.78 NPSR1 (0.73) NPSR1ATMTDP1L3MBTL1PTGIR
SCHEMBL402771 0.77 NPSR1 (0.41) NPSR1ATMTDP1L3MBTL1PTGIR
SCHEMBL17674048 0.73 DHFR (0.42) KMT2AHTTMEN1
SCHEMBL4657473 0.73 ALDH1A1 (0.58) NPSR1L3MBTL1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962830-A2 AZAINDOLE INHIBITORS OF AURORA KINASES SmithKline Beecham Corporation (US) 2008-09-03 EP disclosed
WO-2007076348-A2 AZAINDOLE INHIBITORS OF AURORA KINASES SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed