SCHEMBL5142800

SCHEMBL5142800

Cc1ccc(-n2nc[nH]c2=O)cc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
NPBWR1 P48145 1/20 0.43
XBP1 P17861 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HCAR1 Q9BXC0 1/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
STAT1 P42224 1/20 0.40
GAA P10253 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172956 0.80 ALDH1A1 (0.45) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL8775840 0.78 NPC1 (0.54) ALDH1A1LMNAMAPTCYP1A2NPC1
SCHEMBL19643648 0.73 P2RX7 (0.32) ALDH1A1SMN1; SMN2MAPTHTTNPC1
SCHEMBL8682235 0.73 NPC1 (0.42) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL5906335 0.73 ALDH1A1 (0.40) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL5906387 0.72 MGLL (0.44) ALDH1A1SMN1; SMN2MAPTHTTCYP1A2
SCHEMBL30712345 0.72 MGLL (0.47) ALDH1A1NPBWR1MEN1KMT2AGAA
SCHEMBL8977221 0.72 SMN1; SMN2 (0.47) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL16283450 0.72 SMN1; SMN2 (0.43) ALDH1A1SMN1; SMN2MAPTHTTCYP2C19
SCHEMBL19643603 0.72 CYP2C9 (0.40) ALDH1A1SMN1; SMN2MAPTRAB9ANPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060578-A2 3-ARYL-6-ARYL-[1,2,4] TRIAZOLO[3,4-B][1,3,4] THIADIAZOLES AND RELATED COMPOUNDS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2008-05-22 WO disclosed