SCHEMBL5146071

SCHEMBL5146071

COc1ccc(-c2ccc3nc(NC(C)=O)nc(OCC4CC4)c3c2)cc1OC.COc1ccc(-c2ccc3nc(NC(C)=O)nc(OCCN4CCOCC4)c3c2)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 2/20 0.45
KIT P10721 1/20 0.44
NPC1 O15118 1/20 0.43
CFTR P13569 1/20 0.43
PIK3CA P42336 3/20 0.42
PDE4B Q07343 1/20 0.42
KCNH2 Q12809 3/20 0.42
HTR4 Q13639 3/20 0.42
TRIM58 Q8NG06 1/20 0.41
AVPR1B P47901 1/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
PIK3CD O00329 2/20 0.41
PIK3CB P42338 2/20 0.41
PIK3CG P48736 2/20 0.41
HTR2A P28223 1/20 0.40
ADORA2A P29274 2/20 0.40
ABL1 P00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3339979 0.94 KIT (0.48) MAP3K11KITNPC1CFTRPIK3CA
SCHEMBL3337880 0.88 TRIM58 (0.51) PIK3CATRIM58PIK3CDPIK3CBPIK3CG
SCHEMBL5131263 0.86 KCNH2 (0.44) PIK3CAKCNH2HTR4TRIM58HTR2A
SCHEMBL3336361 0.83 MOK (0.51) PIK3CA
SCHEMBL3334893 0.82 MAPK14 (0.49) PIK3CAKCNH2AVPR1BMAPK13MAPK12
SCHEMBL5127444 0.81 AVPR1B (0.39) NPC1PIK3CAKCNH2HTR4TRIM58
SCHEMBL3332780 0.78 ACHE (0.48) KITPIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL3341092 0.78 ACHE (0.48) KITPIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL3340207 0.78 KIT (0.55) KITNPC1ADORA2ALRRK2
SCHEMBL3341513 0.77 ACHE (0.48) KITPIK3CAPIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed