SCHEMBL5146735

SCHEMBL5146735

COc1cc(CC(=O)NCCCc2ccc3c(c2)OCO3)ccc1OCCN

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
MAPK1 P28482 2/20 0.55
CTSD P07339 3/20 0.52
L3MBTL1 Q9Y468 3/20 0.50
HPGD P15428 1/20 0.50
KMT2A Q03164 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5945398 0.89 HDAC1 (0.49) ALDH1A1MAPK1CTSDHPGD
SCHEMBL5945432 0.89 HDAC1 (0.49) ALDH1A1MAPK1CTSDHPGD
SCHEMBL5945444 0.88 L3MBTL1 (0.63) L3MBTL1MTNR1AMTNR1B
SCHEMBL5945497 0.85 NPC1 (0.49) ALDH1A1MAPK1HPGDKMT2A
SCHEMBL2742524 0.84 ALDH1A1 (0.65) ALDH1A1MAPK1CTSDL3MBTL1HPGD
Davasaicin SCHEMBL5145300 0.84 L3MBTL1 (0.54) L3MBTL1MTNR1AMTNR1B
Davasaicin SCHEMBL30295417 0.84 L3MBTL1 (0.54) L3MBTL1MTNR1AMTNR1B
SCHEMBL5945523 0.83 CA1 (0.59) L3MBTL1MTNR1AMTNR1B
Davasaicin SCHEMBL29396042 0.83 L3MBTL1 (0.53) L3MBTL1MTNR1AMTNR1B
SCHEMBL5945440 0.82 L3MBTL1 (0.55) L3MBTL1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697303-A4 CATALYTIC HYDROGENATION OF NITRILES TO PRODUCE CAPSAICINOID DERIVATIVES AND AMINE COMPOUNDS, AND METHODS FOR PURIFIYING AND OBTAINING THE POLYMORPHS THEREOF STIEFEL LABORATORIES (US) 2007-07-04 EP disclosed
EP-1697303-A1 CATALYTIC HYDROGENATION OF NITRILES TO PRODUCE CAPSAICINOID DERIVATIVES AND AMINE COMPOUNDS, AND METHODS FOR PURIFIYING AND OBTAINING THE POLYMORPHS THEREOF STIEFEL LABORATORIES, INC. (US) 2006-09-06 EP disclosed
US-20060047171-A1 Catalytic hydrogenation of nitriles to produce capsaicinoid derivatives and amine compounds, and methods for purifying and obtaining the polymorphs thereof STIEFEL LABORATORIES, INC. 2006-03-02 US disclosed
WO-2005068414-A1 CATALYTIC HYDROGENATION OF NITRILES TO PRODUCE CAPSAICINOID DERIVATIVES AND AMINE COMPOUNDS, AND METHODS FOR PURIFIYING AND OBTAINING THE POLYMORPHS THEREOF STIEFEL LABORATORIES, INC. (US) 2005-07-28 WO disclosed
EP-0525360-B1 Novel phenylacetamide derivatives and processes for the preparation thereof KOREA RES INST CHEM TECH (KR) 1998-03-25 EP disclosed
US-5242944-A Analgesics or antiinflammatory agents KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1993-09-07 US disclosed
EP-0525360-A2 Novel phenylacetamide derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1993-02-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060047171-A1 Catalytic hydrogenation of nitriles to produce capsaicinoid derivatives and amine compounds, and methods for purifying and obtaining the polymorphs thereof HPD, HNMT, PRPH ALDH1A1 1137/4885MAPK1 2074/4885CTSD 823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.