SCHEMBL5149885

SCHEMBL5149885

O=C(NCCc1ccc(Cl)c(F)c1[N+](=O)[O-])C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
GLA P06280 1/20 0.44
ALOX12 P18054 1/20 0.44
MAPT P10636 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GSTO1 P78417 1/20 0.41
MTNR1A P48039 3/20 0.39
MTNR1B P49286 2/20 0.39
TP53 P04637 1/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9899292 0.75 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1HPGDGLAALOX12
SCHEMBL5152089 0.74 TAAR1 (0.38) SMN1; SMN2ALDH1A1HPGDMAPTNPC1
SCHEMBL5874016 0.73 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1HPGDGLAALOX12
SCHEMBL5855895 0.72 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1HPGDGLAALOX12
SCHEMBL6435988 0.72 TRPV1 (0.60) ALDH1A1HPGDNPC1RAB9AMEN1
SCHEMBL7752152 0.71 CYP1A2 (0.35) SMN1; SMN2HPGDMAPTNPC1RAB9A
SCHEMBL5941728 0.71 TRPV1 (0.58) NPC1RAB9AMTNR1AMTNR1BTP53
SCHEMBL6539895 0.70 KMT2A (0.49) SMN1; SMN2ALDH1A1HPGDGLAALOX12
SCHEMBL5149879 0.70 PDK1 (0.37) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL24826413 0.69 KMT2A (0.46) SMN1; SMN2ALDH1A1HPGDMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1617807-A4 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF ORTHO MCNEIL PHARM INC (US) 2007-02-21 EP disclosed
EP-1617807-A2 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF Ortho-McNeil Pharmaceuticals, Inc. (US) 2006-01-25 EP disclosed
WO-2004096134-A2 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF ORTHO-MCNEIL PHARMACEUTICALS, INC. (US) 2004-11-11 WO disclosed