SCHEMBL5152089

SCHEMBL5152089

NCCc1ccc(Cl)c(F)c1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.38
LMNA P02545 2/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TSHR P16473 2/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
HIF1A Q16665 1/20 0.34
PNMT P11086 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11303709 0.77 ALDH1A1 (0.48) LMNAALDH1A1HPGDMAPTNPC1
SCHEMBL31730954 0.75 TAAR1 (0.48) TAAR1PNMTTDP1
SCHEMBL23152122 0.74 ALDH1A1 (0.44) LMNAALDH1A1HPGDMAPTNPC1
SCHEMBL5149885 0.74 SMN1; SMN2 (0.44) ALDH1A1HPGDMAPTNPC1TP53
SCHEMBL7752152 0.72 CYP1A2 (0.35) LMNAHPGDMAPTNPC1TP53
Hydrochloric Acid SCHEMBL23304051 0.70 TAAR1 (0.44) TAAR1MAPTPNMTHSD17B10TDP1
SCHEMBL25171482 0.70 PTGER4 (0.41) LMNAALDH1A1HPGDMAPTNPC1
SCHEMBL7878527 0.70 GPR35 (0.44) ALDH1A1HPGDTP53SMN1; SMN2TSHR
SCHEMBL24492363 0.70 TAAR1 (0.46) TAAR1ALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL11369484 0.70 HSD17B10 (0.56) TAAR1ALDH1A1HSD17B10TDP1VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1617807-A4 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF ORTHO MCNEIL PHARM INC (US) 2007-02-21 EP disclosed
EP-1617807-A2 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF Ortho-McNeil Pharmaceuticals, Inc. (US) 2006-01-25 EP disclosed
WO-2004096134-A2 SUBSTITUTED 1,4-DIAZEPINES AND USES THEREOF ORTHO-MCNEIL PHARMACEUTICALS, INC. (US) 2004-11-11 WO disclosed