SCHEMBL5150107

SCHEMBL5150107

CCc1c(C)cccc1NCCc1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.47
MTNR1A P48039 2/20 0.45
CA12 O43570 2/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
MAPT P10636 3/20 0.41
HTT P42858 2/20 0.41
ALDH1A1 P00352 5/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
RECQL P46063 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7217415 0.84 NQO2 (0.56) NQO2MTNR1ACA12CA4CA7
SCHEMBL13533413 0.72 NQO2 (0.50) NQO2MTNR1AMAPTHTTALDH1A1
SCHEMBL8414964 0.72 MAPT (0.47) MAPTHTTALDH1A1TSHRHSD17B10
SCHEMBL19122441 0.71 MAPT (0.43) MAPTHTTALDH1A1TSHRHSD17B10
SCHEMBL8858591 0.71 NQO2 (0.58) NQO2MTNR1ACA12CA4CA9
SCHEMBL30420224 0.71 MTNR1A (0.54) NQO2MTNR1AMAPTHTTALDH1A1
SCHEMBL28519744 0.70 MEN1 (0.63) NQO2MTNR1AALDH1A1HSD17B10KDM4E
Ammonia Solution, Strong SCHEMBL9730743 0.70 MAPT (0.42) MAPTHTTALDH1A1TSHRHSD17B10
SCHEMBL606293 0.70 MTNR1A (0.63) NQO2MTNR1AHTTALDH1A1KDM4E
SCHEMBL8794788 0.69 HPGD (0.64) NQO2MTNR1ACA12CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664013-A4 CALCILYTIC COMPOUNDS GLAXO GROUP LTD (GB) 2007-03-14 EP disclosed
EP-1664013-A1 CALCILYTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2006-06-07 EP disclosed
WO-2005030749-A1 CALCILYTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2005-04-07 WO disclosed