SCHEMBL5152136

SCHEMBL5152136

CC(=O)O[C@H]1CCCN1COc1ccc(C(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.42
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
TSHR P16473 2/20 0.40
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTGER4 P35408 5/20 0.40
PTGER2 P43116 2/20 0.39
PKM P14618 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5149767 0.88 KDM4E (0.48) HRH3ALDH1A1TSHRMAPK1KDM4E
SCHEMBL5152988 0.76 KDM4E (0.51) HRH3ALDH1A1KDM4E
SCHEMBL5149764 0.76 KDM4E (0.51) HRH3ALDH1A1KDM4E
SCHEMBL5152354 0.75 KDM4E (0.50) HRH3ALDH1A1KDM4E
SCHEMBL27971258 0.73 ALDH1A1 (0.42) HRH3ALDH1A1
SCHEMBL2087912 0.71 HRH3 (0.67) HRH3
SCHEMBL6959951 0.70 CHRNB2 (0.44) ALDH1A1L3MBTL1PTGER4PTGER2
SCHEMBL14440405 0.70 ALDH1A1 (0.41) ALDH1A1L3MBTL1
SCHEMBL27894922 0.70 ALDH1A1 (0.41) ALDH1A1L3MBTL1
SCHEMBL4654745 0.69 PARP15 (0.45) ALDH1A1TSHRMAPK1USP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179819-B2 VLA-4 inhibitor compounds DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-02-20 US disclosed
US-20040229858-A1 VLA-4 inhibitor compounds DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2004-11-18 US disclosed
US-6756378-B2 BENZYL -UREA, -THIOUREA, OR -GUANIDINE DERIVATIVES THAT INHIBIT THE BINDING OF LIGANDS TO ALPHA 4 BETA 1 INTEGRIN (VLA-4) PHARMACOPEIA DRUG DISCOVERY, INC. 2004-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229858-A1 VLA-4 inhibitor compounds VCAM1, ICAM1, ITGB4 HRH3 1869/4885ALDH1A1 135/4885L3MBTL1 503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.