SCHEMBL5157050

SCHEMBL5157050

CN1CCC(CN2C[C@H](O)C[C@@H]2C(=O)NC23CC4CC(CC(C4)C2)C3)CC1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 10/20 0.44
KDM4E B2RXH2 1/20 0.43
EPHX1 P07099 10/20 0.42
HSD11B1 P28845 1/20 0.39
TSHR P16473 1/20 0.39
CNR2 P34972 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502473 0.88 EPHX1 (0.46) EPHX2EPHX1HSD11B1TSHRCNR2
SCHEMBL6508426 0.85 EPHX1 (0.52) EPHX2EPHX1HSD11B1TSHRCNR2
SCHEMBL5157056 0.79 HSD11B1 (0.53) EPHX2HSD11B1CNR2
SCHEMBL5157962 0.79 EPHX2 (0.46) EPHX2KDM4EEPHX1HSD11B1TSHR
SCHEMBL5158943 0.72 TSHR (0.57) EPHX2EPHX1HSD11B1TSHRCNR2
SCHEMBL6504693 0.70 EPHX1 (0.53) EPHX2EPHX1HSD11B1TSHR
SCHEMBL6507024 0.68 HSD11B1 (0.44) EPHX2HSD11B1
SCHEMBL5160293 0.66 HSD11B1 (0.55) EPHX2KDM4EEPHX1HSD11B1TSHR
SCHEMBL6502476 0.66 HSD11B1 (0.57) EPHX2EPHX1HSD11B1CNR2
SCHEMBL6503334 0.65 ALDH1A1 (0.42) KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745019-A1 NOVEL COMPOUNDS OF PROLINE AND MORPHOLINE DERIVATIVES PFIZER INC. (US) 2007-01-24 EP disclosed
WO-2005108359-A1 NOVEL COMPOUNDS OF PROLINE AND MORPHOLINE DERIVATIVES PFIZER INC. (US) 2005-11-17 WO disclosed