SCHEMBL5157641

SCHEMBL5157641

CN(C)C1(c2ccccc2)CCC(NC(=O)CCC(=O)N2CCC(O)(c3cccc(C(F)(F)F)c3)CC2)CC1.O=C(O)CCCC(=O)N1CCc2ccccc2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.43
OPRL1 P41146 9/20 0.43
CHRM4 P08173 1/20 0.42
CCR2 P41597 4/20 0.40
KCNH2 Q12809 2/20 0.40
OPRK1 P41145 3/20 0.37
TACR1 P25103 1/20 0.37
SIGMAR1 Q99720 2/20 0.37
ABCB11 O95342 1/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
THPO P40225 1/20 0.37
MTOR P42345 1/20 0.37
EBP Q15125 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206307 0.90 OPRM1 (0.52) OPRM1OPRL1CHRM4CCR2KCNH2
SCHEMBL208749 0.81 CCR2 (0.45) OPRM1OPRL1CHRM4CCR2KCNH2
SCHEMBL4084332 0.72 OPRM1 (0.43) OPRM1OPRL1CCR2KCNH2
SCHEMBL206892 0.72 ALDH1A1 (0.48) OPRM1OPRL1CYP3A4CYP2D6PKM
SCHEMBL207055 0.70 OPRM1 (0.57) OPRM1OPRL1CCR2KCNH2SIGMAR1
SCHEMBL206135 0.69 OPRM1 (0.62) OPRM1OPRL1SMN1; SMN2
SCHEMBL207493 0.68 TSHR (0.47) OPRM1OPRL1CHRM4CYP3A4TSHR
SCHEMBL207753 0.68 OPRM1 (0.53) OPRM1OPRL1SIGMAR1
SCHEMBL4072403 0.66 HPGD (0.70) TP53CYP3A4CYP2D6TSHRMAPK1
SCHEMBL3139132 0.65 OPRL1 (0.61) OPRM1OPRL1CHRM4OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536323-A 2007-12-13 JP claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed