SCHEMBL5157777

SCHEMBL5157777

C[Si](C)(C)CCOC(=O)[C@H](Cc1cc(-c2ccc(OCc3ccccc3)c(C[C@H](N)C(=O)OCc3ccccc3)c2)ccc1OCc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CTSK P43235 2/20 0.40
CTSL P07711 2/20 0.40
CTSS P25774 2/20 0.40
CTSB P07858 1/20 0.40
ITGB3 P05106 5/20 0.40
TYR P14679 2/20 0.40
ITGAV P06756 1/20 0.40
IL1RN P18510 1/20 0.39
NMBR P28336 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
ITGA2B P08514 4/20 0.38
TACR1 P25103 1/20 0.38
MBTPS1 Q14703 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5571043 0.99 NOS1 (0.40) NOS1SMN1; SMN2CTSKCTSLCTSS
Hydrochloric Acid SCHEMBL1021511 0.99 NOS1 (0.40) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479149 0.96 NOS1 (0.40) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479144 0.96 ITGB3 (0.41) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479142 0.95 NOS1 (0.38) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479140 0.95 NOS1 (0.38) NOS1SMN1; SMN2CTSKCTSLCTSS
Hydrochloric Acid SCHEMBL1855025 0.94 NOS1 (0.38) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL14497717 0.94 CTSL (0.44) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479152 0.93 NOS1 (0.36) NOS1SMN1; SMN2CTSKCTSLCTSS
SCHEMBL13479143 0.93 GSTP1 (0.40) NOS1SMN1; SMN2CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515983-B1 ANTIBACTERIAL AMIDE MACROCYCLES AICURIS GMBH & CO KG (DE) 2007-02-21 EP disclosed
EP-1526896-A1 ANTIBACTERIAL ESTER MACROCYCLES Bayer HealthCare AG (DE) 2005-05-04 EP disclosed
WO-2004012816-A1 ANTIBACTERIAL ESTER MACROCYCLES BAYER HEALTHCARE AG (DE) 2004-02-12 WO disclosed