SCHEMBL5158010

SCHEMBL5158010

CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)CCC(=O)NCCc2cccc(F)c2)CC1.Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)N3CC=C(c4ccccc4)CC3)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.40
OPRD1 P41143 6/20 0.40
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
SIGMAR1 Q99720 3/20 0.36
CNR1 P21554 2/20 0.35
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5158319 0.88 YAP1 (0.34) OPRM1OPRD1SIGMAR1KDM4EALDH1A1
SCHEMBL205784 0.86 MEN1 (0.49) OPRM1MAPTLMNAHTTKMT2A
SCHEMBL207973 0.85 CNR1 (0.46) OPRM1OPRD1MAPTKMT2ASIGMAR1
SCHEMBL205169 0.84 SIGMAR1 (0.41) MAPTLMNAHTTNPSR1KMT2A
SCHEMBL5154785 0.82 KMT2A (0.36) OPRM1OPRD1MAPTLMNAHTT
SCHEMBL207488 0.82 MEN1 (0.47) OPRM1MAPTLMNAHTTNPSR1
SCHEMBL206590 0.79 MEN1 (0.47) OPRM1MAPTLMNAHTTNPSR1
SCHEMBL206160 0.79 ALDH1A1 (0.49) OPRM1OPRD1MAPTKMT2AMEN1
SCHEMBL208300 0.79 LMNA (0.50) LMNAKMT2AMEN1CNR1TP53
SCHEMBL207909 0.78 HDAC3 (0.45) OPRM1OPRD1LMNAKMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP disclosed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO disclosed