SCHEMBL5159455

SCHEMBL5159455

Cc1nc(NC(C)(C)C)sc1C(=C=O)CN(C)C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
NPC1 O15118 4/20 0.35
CRHR1 P34998 3/20 0.34
POLB P06746 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PIK3CG P48736 1/20 0.34
RAB9A P51151 2/20 0.33
TP53 P04637 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DHODH Q02127 1/20 0.33
HPGD P15428 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
LCK P06239 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5159025 0.85 L3MBTL1 (0.45) ALDH1A1NPC1CRHR1POLBL3MBTL1
SCHEMBL5165151 0.82 MAPK14 (0.40) ALDH1A1NPC1CRHR1POLBL3MBTL1
SCHEMBL5164166 0.81 RAB9A (0.37) ALDH1A1NPC1POLBL3MBTL1RAB9A
SCHEMBL6158103 0.78 NPC1 (0.40) ALDH1A1NPC1CRHR1L3MBTL1RAB9A
SCHEMBL5164299 0.77 ALDH1A1 (0.61) ALDH1A1NPC1CRHR1L3MBTL1PIK3CG
SCHEMBL5159325 0.77 RAB9A (0.56) ALDH1A1NPC1POLBRAB9ATP53
SCHEMBL5161599 0.76 ALDH1A1 (0.35) ALDH1A1HPGD
SCHEMBL5164158 0.75 NPC1 (0.58) ALDH1A1NPC1L3MBTL1RAB9AHTT
SCHEMBL5159300 0.74 NPC1 (0.30) NPC1
SCHEMBL5162743 0.73 NPC1 (0.67) ALDH1A1NPC1RAB9AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756098-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Cyclacel Limited (GB) 2007-02-28 EP disclosed
WO-2005116025-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS CYCLACEL LIMITED (GB) 2005-12-08 WO disclosed