SCHEMBL5161599

SCHEMBL5161599

Cc1nc(N(C)C)sc1C(=C=O)CN(C)C

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5164166 0.87 RAB9A (0.37) ALDH1A1HPGD
SCHEMBL5165104 0.87
SCHEMBL5159300 0.80 NPC1 (0.30)
SCHEMBL5162589 0.79 CRHR1 (0.34)
SCHEMBL5164151 0.79 ADORA2A (0.44) ALDH1A1HPGD
SCHEMBL5159248 0.79 PTGS2 (0.37) ALDH1A1
SCHEMBL6653278 0.79 KMT2A (0.32) ALDH1A1HPGD
SCHEMBL5159025 0.79 L3MBTL1 (0.45) ALDH1A1HPGD
SCHEMBL5165151 0.77 MAPK14 (0.40) ALDH1A1HPGD
SCHEMBL5163544 0.77 CYP1A2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756098-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Cyclacel Limited (GB) 2007-02-28 EP disclosed
WO-2005116025-A2 2-SUBSTITUTED-4-HETEROARYL-PYRIMIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISORDERS CYCLACEL LIMITED (GB) 2005-12-08 WO disclosed