SCHEMBL5161641

SCHEMBL5161641

CC(Oc1ccccc1)C(=O)NC1CCC(Cc2cccc(Cl)c2)(N(C)C)CC1.Cc1ccc(CC2(N(C)C)CCC(NC(=O)COCc3ccccc3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
GHSR Q92847 6/20 0.39
TSHR P16473 1/20 0.37
MCHR1 Q99705 3/20 0.37
FFAR2 O15552 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2984800 0.88 ALDH1A1 (0.48) ALDH1A1MAPTGHSRTSHRFFAR2
SCHEMBL2987025 0.86 SIGMAR1 (0.47) MCHR1SIGMAR1EPHX2
SCHEMBL2982852 0.84 TSHR (0.50) ALDH1A1MAPTTSHR
SCHEMBL2985875 0.83 OPRM1 (0.46) ALDH1A1TSHREPHX2
SCHEMBL5158393 0.82 TSHR (0.38) ALDH1A1GHSRTSHRSIGMAR1
SCHEMBL2976914 0.82 TSHR (0.49) ALDH1A1MAPTGHSRTSHREPHX2
SCHEMBL2985408 0.81 MEN1 (0.47) ALDH1A1MCHR1SIGMAR1
SCHEMBL2985406 0.81 TSHR (0.54) MAPTGHSRTSHR
SCHEMBL2983707 0.79 POLB (0.53) MCHR1SIGMAR1EPHX2
SCHEMBL2989322 0.78 MEN1 (0.48) MAPTTSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536322-A 2007-12-13 JP claimed
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP claimed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO claimed